opioid antagonist उदाहरण वाक्य
उदाहरण वाक्य
- It is still rarely used in medicine in some countries, although it has largely been replaced by more effective respiratory stimulants such as doxapram and specific opioid antagonists such as naloxone.
- Naltrexone is known as an opioid antagonist, a drug that blocks the effects of alcohol on certain chemicals in the brain that normally respond to it, including those that cause pleasurable feelings.
- The effects of morphine can be countered with opioid antagonists such as naloxone and naltrexone; the development of tolerance to morphine may be inhibited by NMDA antagonists such as ketamine or dextromethorphan.
- Some studies using SSRIs have observed that opioid antagonists appear to reduce the urge to steal and mute the " rush " typically experienced immediately after stealing by some subjects suffering from kleptomania.
- The substitution of certain bulky groups on nitrogen 17 converts an opioid agonist into an opioid antagonist, the most important of which is naloxone, a non-selective opioid antagonist with no opioid agonist properties whatsoever.
- The substitution of certain bulky groups on nitrogen 17 converts an opioid agonist into an opioid antagonist, the most important of which is naloxone, a non-selective opioid antagonist with no opioid agonist properties whatsoever.
- A third bill, which has gained little traction elsewhere, would provide immunity from prosecution for anyone who administers prescription drugs known as " opioid antagonists " to reverse the effects of a heroin or opium overdose.
- The compound has relatively little opioid activity in its own right, but is a useful intermediate which can be used to produce both opioid antagonists such as nalorphine, and also potent opioid agonists such as N-phenethylnormorphine.
- Propiram exhibits weak opioid antagonist activity on the mu receptor quite a bit weaker than its agonist effects and the effect on kappa and delta opioid, sigma receptors, or the NMDA system are not well understood.
- If laxatives are insufficiently effective ( which is often the case ), opioid formulations or regimens that include a peripherally-selective opioid antagonist, such as methylnaltrexone bromide, naloxegol, alvimopan, or naloxone ( as in oxycodone / naloxone ), may be tried.